Designed covalent allosteric modulators: an emerging paradigm in drug discovery-Reference-Cited by-同舟云学术

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Designed covalent allosteric modulators: an emerging paradigm in drug discovery

Published:2017-02 Issue:2 Volume:22 Page:447-453
ISSN:1359-6446
Container-title:Drug Discovery Today
language:en
Short-container-title:Drug Discovery Today

Author:

Lu Shaoyong,Zhang Jian

Funder

National Basic Research Program of China (973 Program)

National Natural Science Foundation of China

Shanghai Health and Family Planning Commission

Publisher

Elsevier BV

Subject

Drug Discovery,Pharmacology

Reference60 articles.

1. Targeted covalent inhibitors for drug design;Baillie;Angew. Chem. Int. Ed. Engl.,2016

2. A potentiator of orthosteric ligand activity at GLP-1R acts via covalent modification;Nolte;Nat. Chem. Biol.,2014

3. Targeting transcriptional addictions in small cell lung cancer with a covalent CDK7 inhibitor;Christensen;Cancer Cell,2014

4. Dissecting allosteric effects of activator–coactivator complexes using a covalent small molecule ligand;Wang;Proc. Natl. Acad. Sci. U. S. A.,2014

5. Clickable photoaffinity ligands for metabotropic glutamate receptor 5 based on select acetylenic negative allosteric modulators;Gregory;ACS Chem. Biol.,2016

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