Skin delivery potency and antitumor activities of temozolomide ester prodrugs

Author:

Suppasansatorn Panassaya,Wang Guocheng,Conway Barbara R.,Wang Weidong,Wang Yongfeng

Publisher

Elsevier BV

Subject

Cancer Research,Oncology

Reference29 articles.

1. Comparison of cytotoxicity in vitro of temozolomide and dacarbazine, prodrugs of 3-methyl-(triazen-1-yl)imidazole-4-carboxamide;Tsang;Cancer Chemother. Pharmacol.,1991

2. Antitumour imidazotetrazines XXVIII 3-methyladenine DNA glycosylase activity in cell lines sensitive and resistant to temozolomide;Deans;Cancer Lett.,1992

3. Antitumour activity and pharmacokinetics in mice of 8-carmaboyl-3-methyl-imidazo[5,1 d]-1,2,3,5-tetrazin-4(3H)-one (CCRG 81045; M&B 39831), a novel drug with potential as an alternative to dacarbazine;Stevens;Cancer Res.,1987

4. Activity of temozolomide against human tumour colony-forming units;Raymond;Clin. Cancer Res.,1997

5. Temozolomide: a review of its use in the treatment of malignant gliomas, malignant melanoma and other advanced cancers;Darkes;Am. J. Cancer,2002

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