Troubleshooting problems with in vitro screening of drugs for QT interval prolongation using HERG K+ channels expressed in mammalian cell lines and Xenopus oocytes
Author:
Publisher
Elsevier BV
Subject
Pharmacology,Toxicology
Reference71 articles.
1. Disease-associated mutations in KCNE potassium channel subunits (MiRPs) reveal promiscuous disruption of multiple currents and conservation of mechanism;Abbott;FASEB Journal,2002
2. MiRP1 forms IKr potassium channels with HERG and is associated with cardiac arrhythmia;Abbott;Cell,1999
3. Long-term exposure to retinoic acid induces the expression of IRK1 channels in HERG channel-endowed neuroblastoma cells;Arcangeli;Biochemical and Biophysical Research Communications,1998
4. HERG- and IRK-like inward rectifier currents are sequentially expressed during neuronal development of neural crest cells and their derivatives;Arcangeli;European Journal of Neuroscience,1997
5. Modulation of HERG current and herg gene expression during retinoic acid treatment of human neuroblastoma cells: Potentiating effects of BDNF;Arcangeli;Journal of Neurobiology,1999
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