Synthesis of tubuphenylalanine and epi-tubuphenylalanine via regioselective aziridine ring opening with carbon nucleophiles followed by hydroboration-oxidation of 1,1-substituted amino alkenes-Reference-Cited by-同舟云学术

Synthesis of tubuphenylalanine and epi-tubuphenylalanine via regioselective aziridine ring opening with carbon nucleophiles followed by hydroboration-oxidation of 1,1-substituted amino alkenes

Published:2018-11 Issue:48 Volume:74 Page:6946-6953
ISSN:0040-4020
Container-title:Tetrahedron
language:en
Short-container-title:Tetrahedron

Author:

Reddy Ramesh B.,Dudhe Premansh,Chauhan Priyanka,Sengupta Sagnik,Chelvam Venkatesh

Funder

Department of Science and Technology

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference46 articles.

1. Microtubules as a target for anticancer drugs

2. Mechanism of Action of Tubulysin, an Antimitotic Peptide from Myxobacteria

3. Total Synthesis and Biological Evaluation of Natural and Designed Tubulysins

4. Improved Total Synthesis of Tubulysins and Design, Synthesis, and Biological Evaluation of New Tubulysins with Highly Potent Cytotoxicities against Cancer Cells as Potential Payloads for Antibody–Drug Conjugates

5. The Total Synthesis of Tubulysin D

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3. Synthesis of tubuvaline (Tuv) fragment of tubulysin via diastereoselective dihydroxylation of homoallylamine;Synthetic Communications;2020-12-07

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