Me3SiCl-promoted intramolecular cyclization of aromatic compounds tethered with N,O-acetals leading to the facile preparation of 1,4-benzodiazepine skeletons-Reference-Cited by-同舟云学术

Me3SiCl-promoted intramolecular cyclization of aromatic compounds tethered with N,O-acetals leading to the facile preparation of 1,4-benzodiazepine skeletons

Published:2010-11 Issue:46 Volume:66 Page:8837-8845
ISSN:0040-4020
Container-title:Tetrahedron
language:en
Short-container-title:Tetrahedron

Author:

Sakai Norio,Watanabe Akimasa,Ikeda Reiko,Nakaike Yumi,Konakahara Takeo

Funder

Ministry of Education, Culture, Sports, Science and Technology

Japan Private School Promotion Foundation

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference57 articles.

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2. The Combinatorial Synthesis of Bicyclic Privileged Structures or Privileged Substructures

3. Comparative Quantitative Structure−Activity Relationship Studies (QSAR) on Non-Benzodiazepine Compounds Binding to Benzodiazepine Receptor (BzR)

4. For selected papers, see:

5. A simple route to tetrahydro-1,4-benzodiazepin-3-ones bearing diverse N1, N4, and C10 functionalization

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