A natural compound, aristoyagonine, is identified as a potent bromodomain inhibitor by mid-throughput screening-Reference-Cited by-同舟云学术

A natural compound, aristoyagonine, is identified as a potent bromodomain inhibitor by mid-throughput screening

Published:2018-09 Issue:2 Volume:503 Page:882-887
ISSN:0006-291X
Container-title:Biochemical and Biophysical Research Communications
language:en
Short-container-title:Biochemical and Biophysical Research Communications

Author:

Kim Young Hun,Kim Minsung^ORCID,Yoo Miyoun,Kim Ji Eun,Lee Heung Kyoung,Heo Jung-Nyoung,Lee Chong Ock,Yoo Minjin,Jung Kwan-Young,Yun Chang-Soo,Moon Sung Woong,Chang Hye Kyung,Chung Chul-Woong,Pyo Suhkneung^ORCID,Choi Sang Un,Park Chi Hoon^ORCID

Funder

KRICT

Publisher

Elsevier BV

Subject

Cell Biology,Molecular Biology,Biochemistry,Biophysics

Reference27 articles.

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2. The bromodomain protein Brd4 is a positive regulatory component of P-TEFb and stimulates RNA polymerase II-dependent transcription;Jang;Mol. Cell,2005

3. The Brd4 extraterminal domain confers transcription activation independent of pTEFb by recruiting multiple proteins, including NSD3;Rahman;Mol. Cell Biol.,2011

4. NUT midline carcinoma;French;Canc. Genet. Cytogenet.,2010

5. MYC, a downstream target of BRD-NUT, is necessary and sufficient for the blockade of differentiation in NUT midline carcinoma;Grayson;Oncogene,2014

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