Discovery of BET specific bromodomain inhibitors with a novel scaffold-Reference-Cited by-同舟云学术

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Discovery of BET specific bromodomain inhibitors with a novel scaffold

Published:2022-10 Issue: Volume:72 Page:116967
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Pandit Navin,Yoo Miyoun,Hyun Park Tae,Kim Jiin,Mi Kim Seul,Myung Lee Kyu,Kim Yeongrin,Min Bong Seoung,Il Lee Byung,Jung Kwan-Young,Hoon Park Chi

Funder

Ministry of Science, ICT and Future Planning

Korea Research Institute of Chemical Technology

National Research Foundation of Korea

Korea Drug Development Fund

Korea Ministry of Science and ICT

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference25 articles.

1. Functions of bromodomain-containing proteins and their roles in homeostasis and cancer;Fujisawa;Nat Rev Mol Cell Biol,2017

2. Histone recognition and large-scale structural analysis of the human bromodomain family;Filippakopoulos;Cell,2012

3. The bromodomain protein Brd4 is a positive regulatory component of P-TEFb and stimulates RNA polymerase II-dependent transcription;Jang;Mol Cell,2005

4. Structure and ligand of a histone acetyltransferase bromodomain;Dhalluin;Nature,1999

5. The role of human bromodomains in chromatin biology and gene transcription;Sanchez;Curr Opin Drug Discov Devel,2009

Cited by 1 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Crystal structure of [1,2,4]triazolo[4,3-b]pyridazine derivatives as BRD4 bromodomain inhibitors and structure–activity relationship study;Scientific Reports;2023-07-04

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