Substrate selectivity of human cytochrome P450 2C9: importance of residues 476, 365, and 114 in recognition of diclofenac and sulfaphenazole and in mechanism-based inactivation by tienilic acid-Reference-Cited by-同舟云学术

Substrate selectivity of human cytochrome P450 2C9: importance of residues 476, 365, and 114 in recognition of diclofenac and sulfaphenazole and in mechanism-based inactivation by tienilic acid

Published:2003-01 Issue:1 Volume:409 Page:80-91
ISSN:0003-9861
Container-title:Archives of Biochemistry and Biophysics
language:en
Short-container-title:Archives of Biochemistry and Biophysics

Author:

Melet Armelle,Assrir Nadine,Jean Pascale,Pilar Lopez-Garcia Maria,Marques-Soares Cristina,Jaouen Maryse,Dansette Patrick M,Sari Marie-Agnès,Mansuy Daniel

Publisher

Elsevier BV

Subject

Molecular Biology,Biochemistry,Biophysics

Reference63 articles.

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2. Characterization of cDNAs, mRNAs, and proteins related to human liver microsomal cytochrome P-450 S-mephenytoin 4-hydroxylase

3. Cloning and expression of complementary DNAs for multiple members of the human cytochrome P450IIC subfamily

4. Cytochrome P4502C9: an enzyme of major importance in human drug metabolism

5. Diclofenac and Its Derivatives As Tools for Studying Human Cytochromes P450 Active Sites: Particular Efficiency and Regioselectivity of P450 2Cs

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