Tacrolimus: Does direct glucuronidation matter? An analytical and pharmacological perspective

Author:

Tron Camille,Petitcollin Antoine,Verdier Marie-Clémence,Rayar Michel,Beaurepaire Jean-Marie,Boudjema Karim,Bellissant Eric,Lemaitre Florian

Publisher

Elsevier BV

Subject

Pharmacology

Reference5 articles.

1. A high performance liquid chromatography tandem mass spectrometry for the quantification of tacrolimus in human bile in liver transplant recipients;Tron;J. Chromatogr. A,1475

2. Excretion of tacrolimus glucuronides in human bile;Firdaous;Eur. J. Drug Metab. Pharmacokinet.,1997

3. A practical approach to reduce interference due to in-source collision-induced dissociation of acylglucuronides in LC-MS/MS;Mess;Bioanalysis,2011

4. The role of beta-glucuronidase in drug disposition and drug targeting in humans;Sperker;Clin. Pharmacokinet.,1997

5. In vitro investigation of human UDP-glucuronosyltransferase isoforms responsible for tacrolimus glucuronidation: predominant contribution of UGT1A4;Laverdiere;Drug Metab. Dispos.,2011

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1. Predictors of tacrolimus pharmacokinetic variability: current evidences and future perspectives;Expert Opinion on Drug Metabolism & Toxicology;2020-09-01

2. Pharmacogenetics of Membrane Transporters of Tacrolimus in Solid Organ Transplantation;Clinical Pharmacokinetics;2018-11-10

3. Tacrolimus Elimination in Four Patients With aCYP3A5*3/*3 CYP3A4*22/*22Genotype Combination;Pharmacotherapy: The Journal of Human Pharmacology and Drug Therapy;2018-06-27

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