LJNK, an indoline-2,3-dione-based aminopeptidase N inhibitor with promising antitumor potency

Author:

Hou Jinning,Jin Kang,Li Jin,Jiang Yuqi,Li Xiaoyang,Wang Xuejian,Huang Yongxue,Zhang Yingjie,Xu Wenfang

Publisher

Ovid Technologies (Wolters Kluwer Health)

Subject

Cancer Research,Pharmacology (medical),Pharmacology,Oncology

Reference27 articles.

1. Handbook of Proteolytic Enzymes. 2nd ed.;Barrett;Oxford: Elsevier Academic Press,2004

2. Design, synthesis and primary activity evaluation of L-arginine derivatives as amino-peptidase N/CD13 inhibitors;Mou;Bioorg Med Chem,2009

3. Increased APN/CD13 and acid aminopeptidase activities in head and neck squamous cell carcinoma;Perez;Head neck,2009

4. Ontogenic and adult whole body distribution of aminopeptidase N in rat investigated by in vitro autoradiography;Jardinaud;Biochimie,2004

5. Inflammatory bowel diseases: multiple benefits from therapy with dipeptidyl-and alanyl-aminopeptidase inhibitors;Bank;Front Biosci,2007

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