Addressing the Accuracy of Plasma Protein Binding Measurement for Highly Bound Compounds Using the Dilution Method
Author:
Publisher
Springer Science and Business Media LLC
Subject
Pharmaceutical Science
Link
https://link.springer.com/content/pdf/10.1208/s12248-022-00774-2.pdf
Reference25 articles.
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2. Smith DA, Di L, Kerns EH. The effect of plasma protein binding on in vivo efficacy: misconceptions in drug discovery. Nat Rev Drug Discovery. 2010;9(12):929–39. https://doi.org/10.1038/nrd3287.
3. Liu X, Wright M, Hop CECA. Rational use of plasma protein and tissue binding data in drug design. J Med Chem. 2014;57(20):8238–48. https://doi.org/10.1021/jm5007935.
4. Gardiner P, Cox RJ, Grime K. Plasma protein binding as an optimizable parameter for acidic drugs. Drug Metab Dispos. 2019;47(8):865–73. https://doi.org/10.1124/dmd.119.087163.
5. Di L, Breen C, Chambers R, Eckley ST, Fricke R, Ghosh A, et al. Industry perspective on contemporary protein-binding methodologies: considerations for regulatory drug-drug interaction and related guidelines on highly bound drugs. J Pharm Sci. 2017;106(12):3442–52. https://doi.org/10.1016/j.xphs.2017.09.005.
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