Tetrahydropyrazolo[1,5-a]Pyrimidine-3-Carboxamide and N-Benzyl-6′,7′-Dihydrospiro[Piperidine-4,4′-Thieno[3,2-c]Pyran] Analogues with Bactericidal Efficacy against Mycobacterium tuberculosis Targeting MmpL3

Author:

Remuiñán Modesto J.,Pérez-Herrán Esther,Rullás Joaquín,Alemparte Carlos,Martínez-Hoyos María,Dow David J.,Afari Johnson,Mehta Nalini,Esquivias Jorge,Jiménez Elena,Ortega-Muro Fátima,Fraile-Gabaldón María Teresa,Spivey Vickey L.,Loman Nicholas J.,Pallen Mark J.,Constantinidou Chrystala,Minick Douglas J.,Cacho Mónica,Rebollo-López María José,González Carolina,Sousa Verónica,Angulo-Barturen Iñigo,Mendoza-Losana Alfonso,Barros David,Besra Gurdyal S.,Ballell Lluís,Cammack Nicholas

Publisher

Public Library of Science (PLoS)

Subject

Multidisciplinary

Reference25 articles.

1. WHO (2011) Global Tuberculosis Control: WHO report 2011. Geneva: World Health Organization.

2. The population dynamics and control of tuberculosis;C Dye;Science,2010

3. Multidrug- and extensively drug-resistant tuberculosis: an emerging threat. Eur. Respir. Rev;M Berry,2009

4. The challenge of new drug discovery for tuberculosis;A Koul;Nature,2011

5. Drugs for bad bugs: confronting the challenges of antibacterial discovery;DJ Payne;Nature Drug Discovery,2007

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