Human Biodistribution and Dosimetry of 11C-CUMI-101, an Agonist Radioligand for Serotonin-1A Receptors in Brain-Reference-Cited by-同舟云学术

Human Biodistribution and Dosimetry of 11C-CUMI-101, an Agonist Radioligand for Serotonin-1A Receptors in Brain

Published:2011-09-27 Issue:9 Volume:6 Page:e25309
ISSN:1932-6203
Container-title:PLoS ONE
language:en
Short-container-title:PLoS ONE

Author:

Hines Christina S.,Liow Jeih-San,Zanotti-Fregonara Paolo,Hirvonen Jussi,Morse Cheryl,Pike Victor W.,Innis Robert B.

Publisher

Public Library of Science (PLoS)

Subject

Multidisciplinary

Reference11 articles.

1. Anterior pituitary dopamine receptors. Demonstration of interconvertible high and low affinity states of the D-2 dopamine receptor.;DR Sibley;J Biol Chem,1982

2. The functional state of the dopamine receptor in the anterior pituitary is in the high affinity form.;SR George;Endocrinology,1985

3. In vivo vulnerability to competition by endogenous dopamine: comparison of the D₂ receptor agonist radiotracer (-)-N-[¹¹C]propyl-norapomorphine ([¹¹C]NPA) with the D₂ receptor antagonist radiotracer [¹¹C]-raclopride.;R Narendran;Synapse,2004

4. D₂ dopamine receptor internalization prolongs the decrease of radioligand binding after amphetamine: a PET study in a receptor internalization-deficient mouse model.;M Skinbjerg;Neuro Image,2010

5. Synthesis and in vivo evaluation of a novel 5-HT_1A receptor agonist radioligand [O-methyl- ¹¹C]2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-4-methyl-1,2,4-triazine -3,5(2H,4H)dione in nonhuman primates.;JS Kumar;Eur J Nucl Med Mol Imaging,2007

Cited by 14 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Positron Emission Tomography (PET) Imaging Tracers for Serotonin Receptors;Journal of Medicinal Chemistry;2022-08-08

2. Whole-Body PET Imaging in Humans Shows That¹¹C-PS13 Is Selective for Cyclooxygenase-1 and Can Measure the In Vivo Potency of Nonsteroidal Antiinflammatory Drugs;Journal of Nuclear Medicine;2022-07-07

3. Radiotracers for the Central Serotoninergic System;Pharmaceuticals;2022-05-03

4. 11C Dosimetry Scans Should Be Abandoned;Journal of Nuclear Medicine;2020-12-11

5. Hunting for the high‐affinity state of G‐protein‐coupled receptors with agonist tracers: Theoretical and practical considerations for positron emission tomography imaging;Medicinal Research Reviews;2018-11-18