1. Oncology Discovery, Janssen Research & Development, a division of Janssen Pharmaceutica NV, Turnhoutseweg 30, 2340 Beerse, Belgium
2. Laboratory of Biosignaling & Therapeutics, KULeuven Department of Cellular and Molecular Medicine, University of Leuven, Campus Gasthuisberg, O&N1/ Box 901, Herestraat 49, 3000 Leuven, Belgium
3. Computational Sciences, Janssen Research & Development, a division of Janssen Pharmaceutica NV, Turnhoutseweg 30, 2340 Beerse, Belgium
4. Astex Pharmaceuticals, 436 Cambridge Science Park, Milton Road, Cambridge CB4 0QA, U.K.