Aryl Sulfonamides Induce Degradation of Aryl Hydrocarbon Receptor Nuclear Translocator through CRL4DCAF15 E3 Ligase-Reference-Cited by-同舟云学术

Aryl Sulfonamides Induce Degradation of Aryl Hydrocarbon Receptor Nuclear Translocator through CRL4DCAF15 E3 Ligase

Published:2020-11-30 Issue:11 Volume:43 Page:935-944
ISSN:0219-1032
Container-title:Molecules and Cells
language:en
Short-container-title:Mol.Cells

Author:

Kim Sung Ah¹²^ORCID,Jo Seung-Hyun¹²^ORCID,Cho Jin Hwa¹^ORCID,Yu Min Yeong¹²^ORCID,Shin Ho-Chul¹^ORCID,Kim Jung-Ae³²^ORCID,Park Sung Goo¹²^ORCID,Park Byoung Chul¹⁴^ORCID,Kim Sunhong¹⁵⁶^ORCID,Kim Jeong-Hoon¹²^ORCID

Affiliation:

1. Disease Target Structure Research Center, Korea Research Institute of Bioscience and Biotechnology, Daejeon 34141, Korea

2. Department of Functional Genomics, University of Science and Technology, Daejeon 34113, Korea

3. Personalized Genomic Medicine Research Center, Korea Research Institute of Bioscience and Biotechnology, Daejeon 34141, Korea

4. Department of Bio-Analytical Science, University of Science and Technology, Daejeon 34113, Korea

5. Department of Biomolecular Science, University of Science and Technology, Daejeon 34113, Korea

6. Present address: Drug Discovery Center, LG Chem, Ltd., Seoul 07336, Korea

Funder

Ministry of Science, ICT, and Future Planning

Publisher

Korean Society for Molecular and Cellular Biology

Subject

Cell Biology,Molecular Biology,General Medicine

Link

http://pdf.medrang.co.kr/KSMCB/2020/043/KSMCB043-11-04.pdf

Reference39 articles.

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2. Final results of a phase 2, open-label study of indisulam, idarubicin, and cytarabine in patients with relapsed or refractory acute myeloid leukemia and high-risk myelodysplastic syndrome

3. Cullin-RING ubiquitin ligases: global regulation and activation cycles

4. Structural basis of indisulam-mediated RBM39 recruitment to DCAF15 E3 ligase complex

5. Structural Basis and Kinetic Pathway of RBM39 Recruitment to DCAF15 by a Sulfonamide Molecular Glue E7820

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