Design and synthesis of 4,5-diaryl/heteroarylthiophene-2-carboxylic acid derivatives and evaluation of their biological activities-Reference-Cited by-同舟云学术

Design and synthesis of 4,5-diaryl/heteroarylthiophene-2-carboxylic acid derivatives and evaluation of their biological activities

Published:2017-01-01 Issue:1 Volume:23 Page:
ISSN:2191-0197
Container-title:Heterocyclic Communications
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Author:

Arasavelli Ananda Mohan,Raghava Ganapavarapu Sharma Veera,Vidavalur Siddaiah

Abstract

AbstractSynthesis, characterization and biological activity of novel 4,5-diaryl/heteroaryl thiophene-2-carboxylic acid derivatives are described. Aryl/heteroaryl esters were converted to substituted thiophene esters via a Vilsmeier-Haack reaction, which were then hydrolyzed to 4,5-diaryl/heteroaryl thiophene-2-carboxylic acid derivatives

Publisher

Walter de Gruyter GmbH

Subject

Organic Chemistry

Link

https://www.degruyter.com/document/doi/10.1515/hc-2016-0131/pdf

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