Catalytic Aerobic Oxidation of nor-Binaltorphimine (nor-BNI) Analogs without 4,5-Epoxy Bridge Affords a More Selective Ligand for .KAPPA. Opioid Receptor than the Representative .KAPPA. Antagonist nor-BNI-Reference-Cited by-同舟云学术

Catalytic Aerobic Oxidation of nor-Binaltorphimine (nor-BNI) Analogs without 4,5-Epoxy Bridge Affords a More Selective Ligand for .KAPPA. Opioid Receptor than the Representative .KAPPA. Antagonist nor-BNI

Published:2007 Issue:10 Volume:55 Page:1489-1493
ISSN:0009-2363
Container-title:Chemical and Pharmaceutical Bulletin
language:en
Short-container-title:CHEMICAL & PHARMACEUTICAL BULLETIN

Author:

Osa Yumiko¹,Ida Yoshihiro¹,Fujii Hideaki¹,Nemoto Toru¹,Hasebe Ko²,Momen Shinobu²,Mochizuki Hidenori²,Nagase Hiroshi¹

Affiliation:

1. School of Pharmacy, Kitasato University

2. Pharmaceutical Research Laboratories, Toray Industries, Inc.

Publisher

Pharmaceutical Society of Japan

Subject

Drug Discovery,General Chemistry,General Medicine

Link

http://www.jstage.jst.go.jp/article/cpb/55/10/55_10_1489/_pdf

Reference40 articles.

1. μ-, δ-, κ-Opioid receptors and their subtypes. A critical review with emphasis on radioligand binding experiments

2. Minireview: Multiple MU opiate receptors

3. Analgesic potency of TRIMU-5: A mixed μ2 opioid receptor agonists/μ1 opioid receptor antagonist

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