Pharmacology of Antagonism of GPCR
Author:
Affiliation:
1. Department of Physiology, Graduate School of Pharmaceutical Sciences, Kyushu University
2. Integrated Research Institute for Drug Development, College of Pharmacy, Dongguk University-Seoul
Publisher
Pharmaceutical Society of Japan
Subject
Pharmaceutical Science,Pharmacology,General Medicine
Link
https://www.jstage.jst.go.jp/article/bpb/45/6/45_b22-00143/_pdf
Reference35 articles.
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3. 3) Syrovatkina V, Alegre KO, Dey R, Huang X-Y. Regulation, signaling, and physiological functions of G-proteins. J. Mol. Biol., 428, 3850–3868 (2016).
4. 4) Fredriksson R, Lagerström MC, Lundin L-G, Schiöth HB. The G-protein-coupled receptors in the human genome form five main families. Phylogenetic analysis, paralogon groups, and fingerprints. Mol. Pharmacol., 63, 1256–1272 (2003).
5. 5) Masureel M, Zou Y, Picard L-P, van der Westhuizen E, Mahoney JP, Rodrigues JPGLM, Mildorf TJ, Dror RO, Shaw DE, Bouvier M, Pardon E, Steyaert J, Sunahara RK, Weis WI, Zhang C, Kobilka BK. Structural insights into binding specificity, efficacy and bias of a β2AR partial agonist. Nat. Chem. Biol., 14, 1059–1066 (2018).
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