Establishment of a Stable Human Cell Line, HPL-A3, for Use in Reporter Gene Assays of Cytochrome P450 3A Inducers-Reference-Cited by-同舟云学术

Establishment of a Stable Human Cell Line, HPL-A3, for Use in Reporter Gene Assays of Cytochrome P450 3A Inducers

Published:2012 Issue:5 Volume:35 Page:677-685
ISSN:0918-6158
Container-title:Biological and Pharmaceutical Bulletin
language:en
Short-container-title:Biol. Pharm. Bull.

Author:

Sekimoto Masashi¹,Sano Shinsuke¹,Hosaka Takuomi¹,Nemoto Kiyomitsu¹,Degawa Masakuni¹

Affiliation:

1. Department of Molecular Toxicology and Global Center of Excellence Program, School of Pharmaceutical Sciences, University of Shizuoka

Publisher

Pharmaceutical Society of Japan

Subject

Pharmaceutical Science,Pharmacology,General Medicine

Link

https://www.jstage.jst.go.jp/article/bpb/35/5/35_5_677/_pdf

Reference41 articles.

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2. Drugs Behave as Substrates, Inhibitors and Inducers of Human Cytochrome P450 3A4

3. 3) Tachibana T, Kato M, Takano J, Sugiyama Y. Predicting drug–drug interactions involving the inhibition of intestinal CYP3A4 and P-glycoprotein. Curr. Drug Metab., 11, 762–777 (2010).

4. 4) Donato MT, Lahoz A, Castell JV, Gómez-Lechón MJ. Cell lines: a tool for in vitro drug metabolism studies. Curr. Drug Metab., 9, 1–11 (2008).

5. EXPRESSION OF CYTOCHROMES P450, CONJUGATING ENZYMES AND NUCLEAR RECEPTORS IN HUMAN HEPATOMA HepaRG CELLS

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