Boehringer Ingleheim's selective glucocorticoid receptor agonist development candidate: evaluation of WO2010141331, WO2010141332 and WO2010141333
Author:
Publisher
Informa Healthcare
Subject
Drug Discovery,Pharmacology,General Medicine
Link
http://www.tandfonline.com/doi/pdf/10.1517/13543776.2011.581229
Reference12 articles.
1. Inhaled corticosteroids as combination therapy with β-adrenergic agonists in airways disease: present and future
2. New Insights into the Molecular Mechanisms of Corticosteroids Actions
3. X-ray Crystal Structure of the Novel Enhanced-Affinity Glucocorticoid Agonist Fluticasone Furoate in the Glucocorticoid Receptor−Ligand Binding Domain
4. Design and x-ray crystal structures of high-potency nonsteroidal glucocorticoid agonists exploiting a novel binding site on the receptor
5. Dissociated non-steroidal glucocorticoid receptor modulators: an update on new compounds
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