1-(5-Carboxyindazol-1-yl)propan-2-ones as dual inhibitors of cytosolic phospholipase A2α and fatty acid amide hydrolase: bioisosteric replacement of the carboxylic acid moiety-Reference-Cited by-同舟云学术

1-(5-Carboxyindazol-1-yl)propan-2-ones as dual inhibitors of cytosolic phospholipase A2α and fatty acid amide hydrolase: bioisosteric replacement of the carboxylic acid moiety

Published:2016-05-09 Issue:sup1 Volume:31 Page:131-140
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Althaus Jan¹,Hake Theresa¹,Hanekamp Walburga¹,Lehr Matthias¹

Affiliation:

1. Institute of Pharmaceutical and Medicinal Chemistry, University of Münster, Germany

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2016.1178246

Reference22 articles.

1. Phospholipase A2 Enzymes: Physical Structure, Biological Function, Disease Implication, Chemical Inhibition, and Therapeutic Intervention

2. Cytosolic phospholipase A2: physiological function and role in disease

3. Endocannabinoids: synthesis and degradation

4. Fatty Acid Amide Hydrolase: A Gate-Keeper of the Endocannabinoid System

5. CHAPTER 2. Inhibitors of Cytosolic Phospholipase A2α as Anti-inflammatory Drugs

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