Isoxazol-5(2H)-one: a new scaffold for potent human neutrophil elastase (HNE) inhibitors-Reference-Cited by-同舟云学术

Isoxazol-5(2H)-one: a new scaffold for potent human neutrophil elastase (HNE) inhibitors

Published:2017-01-01 Issue:1 Volume:32 Page:821-831
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Vergelli Claudia¹,Schepetkin Igor A.²,Crocetti Letizia¹,Iacovone Antonella¹,Giovannoni Maria Paola¹,Guerrini Gabriella¹,Khlebnikov Andrei I.³⁴,Ciattini Samuele⁵,Ciciani Giovanna¹,Quinn Mark T.²

Affiliation:

1. NEUROFARBA, Sezione di Farmaceutica e Nutraceutica, Università degli Studi di Firenze, Sesto Fiorentino, Italy;

2. Department of Microbiology and Immunology, Montana State University, Bozeman, MT, USA;

3. Department of Biotechnology and Organic Chemistry, Tomsk Polytechnic University, Tomsk, Russia;

4. Department of Chemistry, Altai State Technical University, Barnaul, Russia;

5. Dipartimento di Chimica, Centro di Cristallografia, Università degli Studi di Firenze, Sesto Fiorentino, Italy

Funder

National Institutes of Health

USDA National Institute of Food and Agriculture

Ministry of Education and Science of the Russian Federation

University of Montana

Montana State University

the Ministry of Education and Science of the Russian Federation

U.S. Department of Agriculture

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://tandfonline.com/doi/pdf/10.1080/14756366.2017.1326915

Reference41 articles.

1. Serine proteases of the human immune system in health and disease

2. Neutrophil Elastase, Proteinase 3, and Cathepsin G as Therapeutic Targets in Human Diseases

3. Neutrophil Elastase: Mediator of Extracellular Matrix Destruction and Accumulation

4. The Balancing Act of Neutrophils

Cited by 30 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Exploration of novel human neutrophil elastase inhibitors from natural compounds: Virtual screening, in vitro, molecular dynamics simulation and in vivo study;European Journal of Pharmacology;2024-11

2. Human neutrophil elastase inhibitors: Classification, biological‐synthetic sources and their relevance in related diseases;Fundamental & Clinical Pharmacology;2023-08-23

3. Design and synthesis of thiadiazole-oxadiazole-acetamide derivatives: Elastase inhibition, cytotoxicity, kinetic mechanism, and computational studies;Bioorganic & Medicinal Chemistry;2023-05

4. Continuous Flow Photochemical Synthesis of 3-Methyl-4-arylmethylene Isoxazole-5(4H)-ones through Organic Photoredox Catalysis and Investigation of Their Larvicidal Activity;Catalysts;2023-03-03

5. X-ray structural study of human neutrophil elastase inhibition with a series of azaindoles, azaindazoles and isoxazolones;Journal of Molecular Structure;2023-02