Design, synthesis, molecular modeling and biological evaluation of novel Benzoxazole-Benzamide conjugates <i>via</i> a 2-Thioacetamido linker as potential anti-proliferative agents, VEGFR-2 inhibitors and apoptotic inducers-Reference-Cited by-同舟云学术

Design, synthesis, molecular modeling and biological evaluation of novel Benzoxazole-Benzamide conjugates via a 2-Thioacetamido linker as potential anti-proliferative agents, VEGFR-2 inhibitors and apoptotic inducers

Published:2022-05-30 Issue:1 Volume:37 Page:1587-1599
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Eissa Ibrahim H.¹^ORCID,El-Haggar Radwan²³,Dahab Mohammed A.¹,Ahmed Marwa F.²⁴,Mahdy Hazem A.¹^ORCID,Alsantali Reem I.⁴,Elwan Alaa¹,Masurier Nicolas³^ORCID,Fatahala Samar S.⁵

Affiliation:

1. Pharmaceutical Medicinal Chemistry & Drug Design Department, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo, Egypt

2. Pharmaceutical Chemistry Department, Faculty of Pharmacy, Helwan University, Cairo, Egypt

3. Institut des Biomolécules Max Mousseron (IBMM), UMR 5247, CNRS, Université de Montpellier, ENSCM, Montpellier, France

4. Department of Pharmaceutical Chemistry, College of Pharmacy, Taif University, Taif, Saudi Arabia

5. Pharmaceutical Organic Chemistry Department, Faculty of Pharmacy, Helwan University, Cairo, Egypt

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2022.2081844

Reference70 articles.

1. Protein tyrosine kinase inhibitors: new treatment modalities?

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