Synthesis, molecular modelling and QSAR study of new <i>N-</i>phenylacetamide-2-oxoindole benzensulfonamide conjugates as carbonic anhydrase inhibitors with antiproliferative activity-Reference-Cited by-同舟云学术

Synthesis, molecular modelling and QSAR study of new N-phenylacetamide-2-oxoindole benzensulfonamide conjugates as carbonic anhydrase inhibitors with antiproliferative activity

Published:2022-02-15 Issue:1 Volume:37 Page:701-717
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Said Mona F.¹,George Riham F.¹^ORCID,Petreni Andrea²,Supuran Claudiu T.²^ORCID,Mohamed Nada M.³

Affiliation:

1. Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Cairo, Egypt

2. Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Florence, Italy

3. Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Modern University for Technology and Information MTI, Cairo, Egypt

Funder

Italian Ministry for Education and Science

Ente Cassa di Risparmio di Firenze

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2022.2036137

Reference59 articles.

1. Structure and function of carbonic anhydrases

2. Catalytic Mechanism of α-Class Carbonic Anhydrases: CO2 Hydration and Proton Transfer

3. Carbonic Anhydrase Inhibitors Drug Design

4. Structure-based drug discovery of carbonic anhydrase inhibitors

5. Inhibitory effects and structural insights for a novel series of coumarin-based compounds that selectively target human CA IX and CA XII carbonic anhydrases

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