Design, synthesis, and anti-cancer evaluation of new pyrido[2,3-d]pyrimidin-4(3H)-one derivatives as potential EGFRWT and EGFRT790M inhibitors and apoptosis inducers

Author:

Elzahabi Heba S. A.1ORCID,Nossier Eman S.1,Alasfoury Rania A.1,El-Manawaty May2,Sayed Sara M.3,Elkaeed Eslam B.4,Metwaly Ahmed M.56,Hagras Mohamed7,Eissa Ibrahim H.8ORCID

Affiliation:

1. Pharmaceutical Medicinal Chemistry & Drug Design Department, Faculty of Pharmacy (Girls), Al-Azhar University, Cairo, Egypt

2. Pharmacognosy Department, National Research Centre, Dokki, Cairo, Egypt

3. Biochemistry and Molecular Biology Department, Faculty of Pharmacy (Girls), Al-Azhar University, Cairo, Egypt

4. Department of Pharmaceutical Sciences, College of Pharmacy, AlMaarefa University, Riyadh, Saudi Arabia

5. Pharmacognosy and Medicinal Plants Department, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo, Egypt

6. Biopharmaceutical Products Research Department, Genetic Engineering and Biotechnology Research Institute, City of Scientific Research and Technological Applications (SRTA-City), Alexandria, Egypt

7. Pharmaceutical Organic Chemistry, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo, Egypt

8. Pharmaceutical Medicinal Chemistry & Drug Design Department, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo, Egypt

Funder

Science, Technology & Innovation Funding Authority

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Reference78 articles.

1. WHO. Cancer. Available from: https://www.who.int/news-room/fact-sheets/detail/cancer. (last accessed 13 Jan 2022).

2. Cancer incidence and mortality in Europe, 2004

3. MicroRNAs and their role in environmental chemical carcinogenesis

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