Antihistamines, phenothiazine-based antipsychotics, and tricyclic antidepressants potently activate pharmacologically relevant human carbonic anhydrase isoforms II and VII-Reference-Cited by-同舟云学术

Antihistamines, phenothiazine-based antipsychotics, and tricyclic antidepressants potently activate pharmacologically relevant human carbonic anhydrase isoforms II and VII

Published:2023-03-13 Issue:1 Volume:38 Page:
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Fiorentino Francesco¹^ORCID,Nocentini Alessio²^ORCID,Rotili Dante¹^ORCID,Supuran Claudiu T.²^ORCID,Mai Antonello¹³^ORCID

Affiliation:

1. Department of Drug Chemistry and Technologies, Sapienza University of Rome, Rome, Italy

2. Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, Polo Scientifico, University of Florence, Firenze, Italy

3. Pasteur Institute, Cenci-Bolognetti Foundation, Sapienza University of Rome, Rome, Italy

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2023.2188147

Reference84 articles.

1. How many carbonic anhydrase inhibition mechanisms exist?

2. Multiple Binding Modes of Inhibitors to Carbonic Anhydrases: How to Design Specific Drugs Targeting 15 Different Isoforms?

3. Exploring the multiple binding modes of inhibitors to carbonic anhydrases for novel drug discovery

4. Carbonic anhydrases: novel therapeutic applications for inhibitors and activators

5. Amine- and Amino Acid-Based Compounds as Carbonic Anhydrase Activators

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