Structure activity relationship studies on Amb639752: toward the identification of a common pharmacophoric structure for DGKα inhibitors-Reference-Cited by-同舟云学术

Structure activity relationship studies on Amb639752: toward the identification of a common pharmacophoric structure for DGKα inhibitors

Published:2019-11-05 Issue:1 Volume:35 Page:96-108
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Velnati Suresh¹²,Massarotti Alberto³,Antona Annamaria¹,Talmon Maria⁴,Fresu Luigia Grazia⁴,Galetto Alessandra Silvia¹⁵,Capello Daniela¹,Bertoni Alessandra¹,Mercalli Valentina³,Graziani Andrea⁶⁷,Tron Gian Cesare³,Baldanzi Gianluca¹²

Affiliation:

1. Department of Translational Medicine, University of Piemonte Orientale, Novara, Italy

2. Institute for Research and Cure of Autoimmune Diseases, CAAD, University of Piemonte Orientale, Novara, Italy

3. Department of Pharmaceutical Sciences, University of Piemonte Orientale, Novara, Italy

4. Department of Health Sciences, School of Medicine, University of Piemonte Orientale, Novara, Italy

5. Palliative Care Division, A.S.L., Vercelli, Italy

6. Università Vita-Salute San Raffaele, Milan, Italy

7. Department of Molecular Biotechnology and Health Sciences, Molecular Biotechnology Center, University of Torino, Turin, Italy

Funder

Università del Piemonte Orientale

Telethon Foundation

National Ministry of University and Research PRIN 2017

Consorzio Interuniversitario di Biotecnologie (CIB) bando “Network-CIB: Catalisi dell’Innovazione nelle biotecnologie”

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2019.1684911

Reference43 articles.

1. Diacylglycerol kinases as sources of phosphatidic acid

2. Role of Diacylglycerol Kinases in T Cell Development and Function

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4. Diacylglycerol kinases: Why so many of them?

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