Reprofiling of pyrimidine-based DAPK1/CSF1R dual inhibitors: identification of 2,5-diamino-4-pyrimidinol derivatives as novel potential anticancer lead compounds-Reference-Cited by-同舟云学术

Reprofiling of pyrimidine-based DAPK1/CSF1R dual inhibitors: identification of 2,5-diamino-4-pyrimidinol derivatives as novel potential anticancer lead compounds

Published:2019-12-06 Issue:1 Volume:35 Page:311-324
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Farag Ahmed K.¹^ORCID,Hassan Ahmed H. E.²^ORCID,Ahn Byung Sun³⁴,Park Ki Duk⁴⁵,Roh Eun Joo³⁴

Affiliation:

1. RI Translational Research Team, Division of Applied RI, Korea Institute of Radiological and Medical Sciences (KIRAMS), Seoul, Republic of Korea

2. Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt

3. Chemical Kinomics Research Center, Korea Institute of Science and Technology (KIST), Seoul, Republic of Korea

4. Division of Bio-Medical Science and Technology, KIST School, University of Science and Technology, Seoul, Republic of Korea

5. Convergence Research Center for Diagnosis, Treatment and Care System of Dementia, Korea Institute of Science and Technology (KIST), Seoul, Republic of Korea

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2019.1699554

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4. Design, synthesis and evaluation of alkylphosphocholine-gefitinib conjugates as multitarget anticancer agents

5. A Review on Synthesis, Anticancer and Antiviral Potentials of Pyrimidine Derivatives

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