Fibrate-based N-acylsulphonamides targeting carbonic anhydrases: synthesis, biochemical evaluation, and docking studies-Reference-Cited by-同舟云学术

Fibrate-based N-acylsulphonamides targeting carbonic anhydrases: synthesis, biochemical evaluation, and docking studies

Published:2019-01-01 Issue:1 Volume:34 Page:1051-1061
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Ammazzalorso Alessandra¹,Carradori Simone¹^ORCID,Angeli Andrea²^ORCID,Akdemir Atilla³,De Filippis Barbara¹,Fantacuzzi Marialuigia¹,Giampietro Letizia¹,Maccallini Cristina¹,Amoroso Rosa¹,Supuran Claudiu T.²⁴^ORCID

Affiliation:

1. Department of Pharmacy, “G. d’Annunzio” University of Chieti-Pescara, Chieti, Italy;

2. Laboratorio di Chimica Bioinorganica, Università degli Studi di Firenze, Florence, Italy;

3. Department of Pharmacology, Faculty of Pharmacy, Computer-Aided Drug Discovery Laboratory, Bezmialem Vakif University, Istanbul, Turkey;

4. Neurofarba Department, Section of Pharmaceutical and Nutriceutical Sciences, Università degli Studi di Firenze, Florence, Italy

Funder

FAR funds

Italian Ministry for Instruction, University and Research

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://tandfonline.com/doi/pdf/10.1080/14756366.2019.1611801

Reference57 articles.

1. Sulfonamides and their isosters as carbonic anhydrase inhibitors

2. Sulfonamides and their isosters as carbonic anhydrase inhibitors

3. Sulfonamides as Potential Bioactive Scaffolds

4. N -acylsulfonamides: Synthetic routes and biological potential in medicinal chemistry

5. Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design

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