Discovery of new pyridine-quinoline hybrids as competitive and non-competitive PIM-1 kinase inhibitors with apoptosis induction and caspase 3/7 activation capabilities-Reference-Cited by-同舟云学术

Discovery of new pyridine-quinoline hybrids as competitive and non-competitive PIM-1 kinase inhibitors with apoptosis induction and caspase 3/7 activation capabilities

Published:2023-01-11 Issue:1 Volume:38 Page:
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

El-Miligy Mostafa M. M.¹^ORCID,Abdelaziz Marwa E.¹,Fahmy Salwa M.¹,Ibrahim Tamer M.²,Abu-Serie Marwa M.³,Mahran Mona A.¹,Hazzaa Aly A.¹

Affiliation:

1. Pharmaceutical Chemistry Department, Faculty of Pharmacy, Alexandria University, Alexandria, Egypt

2. Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, Egypt

3. Medical Biotechnology Department, Genetic Engineering and Biotechnology Research Institute (GEBRI, City of Scientific Research and Technological Applications (SRTA-City), Alexandria, Egypt)

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2022.2152810

Reference47 articles.

1. Inhibition of FLT3 and PIM Kinases by EC-70124 Exerts Potent Activity in Preclinical Models of Acute Myeloid Leukemia

2. Insights from Pim1 structure for anti-cancer drug design

3. Using Insights into Pim1 Structure to Design New Anticancer Drugs

4. Pim kinases in cancer: Diagnostic, prognostic and treatment opportunities

5. Medicinal attributes of pyridine scaffold as anticancer targeting agents

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