Dependence on linkers’ flexibility designed for benzenesulfonamides targeting discovery of novel hCA IX inhibitors as potent anticancer agents-Reference-Cited by-同舟云学术

Dependence on linkers’ flexibility designed for benzenesulfonamides targeting discovery of novel hCA IX inhibitors as potent anticancer agents

Published:2022-10-09 Issue:1 Volume:37 Page:2765-2785
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Tawfik Haytham O.¹^ORCID,Belal Amany²³^ORCID,Abourehab Mohammed A. S.⁴⁵^ORCID,Angeli Andrea⁶^ORCID,Bonardi Alessandro⁶,Supuran Claudiu T.⁶^ORCID,El-Hamamsy Mervat H.¹

Affiliation:

1. Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Tanta University, Tanta, Egypt

2. Medicinal Chemistry Department, Faculty of Pharmacy, Beni-Suef University, Beni-Suef, Egypt

3. Department of Pharmaceutical Chemistry, College of Pharmacy, Taif University, Taif, Saudi Arabia

4. Department of Pharmaceutics, Faculty of Pharmacy, Umm Al-Qura University, Makkah, Saudi Arabia

5. Department of Pharmaceutics and Industrial Pharmacy, College of Pharmacy, Minia University, Minia, Egypt

6. Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Sesto Fiorentino, Italy

Funder

Faculty of Pharmacy, Tanta University, and the Deanship of scientific

Umm Al-Qura University

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2022.2130285

Reference77 articles.

1. Genome-wide identification, phylogeny, and expression analysis of the CA gene family in tomato

2. Emerging roles for carbonic anhydrase in mesophyll conductance and photosynthesis

3. Betulin Sulfonamides as Carbonic Anhydrase Inhibitors and Anticancer Agents in Breast Cancer Cells

4. Proton Transport in Cancer Cells: The Role of Carbonic Anhydrases

5. Carbonic anhydrases as targets for medicinal chemistry

Cited by 19 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Fragment-based design and synthesis of coumarin-based thiazoles as dual c-MET/STAT-3 inhibitors for potential antitumor agents;Bioorganic Chemistry;2024-10

2. Unveiling the potential of isatin-grafted phenyl-1,2,3-triazole derivatives as dual VEGFR-2/STAT-3 inhibitors: Design, synthesis and biological assessments;Bioorganic Chemistry;2024-10

3. Novel sulfonamide-tethered Schiff bases as anti-proliferative agents with VEGFR-2 inhibitory activity: Synthesis, biological assessment, and molecular dynamic simulations;Journal of Molecular Structure;2024-08

4. A new framework for novel analogues of pazopanib as potent and selective human carbonic anhydrase inhibitors: Design, repurposing rational, synthesis, crystallographic, in vivo and in vitro biological assessments;European Journal of Medicinal Chemistry;2024-08

5. Rationale design of novel substituted 1,3,5-triazine candidates as dual IDH1(R132H)/ IDH2(R140Q) inhibitors with high selectivity against acute myeloid leukemia: In vitro and in vivo preclinical investigations;Bioorganic Chemistry;2024-08