Novel hits for acetylcholinesterase inhibition derived by docking-based screening on ZINC database-Reference-Cited by-同舟云学术

Novel hits for acetylcholinesterase inhibition derived by docking-based screening on ZINC database

Published:2018-01-01 Issue:1 Volume:33 Page:768-776
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Doytchinova Irini¹²^ORCID,Atanasova Mariyana¹,Valkova Iva¹²,Stavrakov Georgi¹³,Philipova Irena³,Zhivkova Zvetanka¹,Zheleva-Dimitrova Dimitrina¹,Konstantinov Spiro¹,Dimitrov Ivan¹

Affiliation:

1. Faculty of Pharmacy, Medical University of Sofia, Sofia, Bulgaria;

2. Drug Design and Development Lab, Sofia Tech Park, Sofia, Bulgaria;

3. Institute of Organic Chemistry with Centre of Phytochemistry, Bulgarian Academy of Sciences, Sofia, Bulgaria

Funder

Medical Research Council, Medical University of Sofia

Bulgarian National Science Fund

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2018.1458031

Reference55 articles.

1. The Cholinergic Hypothesis of Geriatric Memory Dysfunction

2. On Neurodegenerative Diseases, Models, and Treatment Strategies: Lessons Learned and Lessons Forgotten a Generation Following the Cholinergic Hypothesis

3. Alzheimer’s Disease Therapy: Present and Future Molecules

4. Functional Characteristics of the Oxyanion Hole in Human Acetylcholinesterase

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