Design, synthesis, in vitro antiproliferative activity and apoptosis-inducing studies of 1-(3′,4′,5′-trimethoxyphenyl)-3-(2′-alkoxycarbonylindolyl)-2-propen-1-one derivatives obtained by a molecular hybridisation approach-Reference-Cited by-同舟云学术

Design, synthesis, in vitro antiproliferative activity and apoptosis-inducing studies of 1-(3′,4′,5′-trimethoxyphenyl)-3-(2′-alkoxycarbonylindolyl)-2-propen-1-one derivatives obtained by a molecular hybridisation approach

Published:2018-01-01 Issue:1 Volume:33 Page:1225-1238
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Preti Delia¹,Romagnoli Romeo¹,Rondanin Riccardo¹,Cacciari Barbara¹,Hamel Ernest²,Balzarini Jan³,Liekens Sandra³,Schols Dominique³,Estévez-Sarmiento Francisco⁴,Quintana José⁴,Estévez Francisco⁴

Affiliation:

1. Department of Chemical and Pharmaceutical Sciences, University of Ferrara, Ferrara, Italy;

2. Screening Technologies Branch, Developmental Therapeutics Program, Division of Cancer Treatment and Diagnosis, Frederick National Laboratory for Cancer Research, National Cancer Institute, National Institutes of Health, Frederick, MD, USA;

3. Rega Institute for Medical Research, KU Leuven, Laboratory of Virology and Chemotherapy, Leuven, Belgium;

4. Department of Biochemistry and Molecular Biology, Research Institute in Biomedical and Health Sciences (IUIBS), University of Las Palmas de Gran Canaria (ULPGC), Spain

Funder

“Finanziamento delle attività base di ricerca 2017”

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2018.1493473

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