Synthesis, biological evaluation, and molecular modelling studies of potent human neutrophil elastase (HNE) inhibitors-Reference-Cited by-同舟云学术

Synthesis, biological evaluation, and molecular modelling studies of potent human neutrophil elastase (HNE) inhibitors

Published:2018-01-01 Issue:1 Volume:33 Page:1108-1124
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Giovannoni Maria Paola¹^ORCID,Schepetkin Igor A.²^ORCID,Quinn Mark T.²^ORCID,Cantini Niccolò¹,Crocetti Letizia¹,Guerrini Gabriella¹^ORCID,Iacovone Antonella¹,Paoli Paola³^ORCID,Rossi Patrizia³^ORCID,Bartolucci Gianluca¹^ORCID,Menicatti Marta¹,Vergelli Claudia¹^ORCID

Affiliation:

1. NEUROFARBA, Pharmaceutical and Nutraceutical Section, University of Florence, Sesto Fiorentino, Italy;

2. Department of Microbiology and Immunology, Montana State University, Bozeman, MT, USA;

3. Department of Industrial Engineering, University of Florence, Florence, Italy

Funder

National Institutes of Health

National Institute of Food and Agriculture

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2018.1480615

Reference71 articles.

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4. NSP4, an elastase-related protease in human neutrophils with arginine specificity

5. Neutrophil Elastase, Proteinase 3, and Cathepsin G as Therapeutic Targets in Human Diseases

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