S-substituted 2-mercaptoquinazolin-4(3H)-one and 4-ethylbenzensulfonamides act as potent and selective human carbonic anhydrase IX and XII inhibitors-Reference-Cited by-同舟云学术

S-substituted 2-mercaptoquinazolin-4(3H)-one and 4-ethylbenzensulfonamides act as potent and selective human carbonic anhydrase IX and XII inhibitors

Published:2020-01-01 Issue:1 Volume:35 Page:733-743
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

El-Azab Adel S.¹^ORCID,Abdel-Aziz Alaa A.-M.¹^ORCID,Bua Silvia²,Nocentini Alessio²,AlSaif Nawaf A.¹,Alanazi Mohammed M.¹,El-Gendy Manal A.¹,Ahmed Hany E. A.³⁴,Supuran Claudiu T.²^ORCID

Affiliation:

1. Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh, Saudi Arabia

2. Department of Neurofarba, Sezione di Scienze Farmaceutiche e Nutraceutiche, Università degli Studi di Firenze, Florence, Italy

3. Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Al-Azhar University, Cairo, Egypt

4. Pharmacognosy and Pharmaceutical Chemistry Department, College of Pharmacy, Taibah University, Al-Madinah Al-Munawarah, Saudi Arabia

Funder

King Saud University

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2020.1742117

Reference70 articles.

1. Advances in the structural annotation of human carbonic anhydrases and impact on future drug discovery

2. Carbonic anhydrases: novel therapeutic applications for inhibitors and activators

3. Multiple Binding Modes of Inhibitors to Carbonic Anhydrases: How to Design Specific Drugs Targeting 15 Different Isoforms?

4. Carbonic anhydrase inhibitors as antitumor/antimetastatic agents: a patent review (2008–2018)

5. How many carbonic anhydrase inhibition mechanisms exist?

Cited by 26 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Prominent antidiabetic and anticancer investigation of Scrophularia deserti extract: Integration of experimental and computational approaches;Journal of Molecular Structure;2024-11

2. Synthesis of new sulfonamide derivatives: Investigation of their interactions with carbonic anhydrase and cholinesterase enzymes by in vitro and in silico evaluations;Journal of Molecular Structure;2024-10

3. Chemistry of heterocycles as carbonic anhydrase inhibitors: A pathway to novel research in medicinal chemistry review;Archiv der Pharmazie;2024-04-29

4. Green synthesis of 2‐thioxo‐4‐quinazolinones from 2‐aminobenzamide and isothiocyanates;Vietnam Journal of Chemistry;2024-03-14

5. Identification of thienopyrimidine derivatives tethered with sulfonamide and other moieties as carbonic anhydrase inhibitors: Design, synthesis and anti-proliferative activity;Bioorganic Chemistry;2024-03