Insights into the cellular pharmacological properties of the BET-inhibitor OTX015/MK-8628 (birabresib), alone and in combination, in leukemia models

Author:

Astorgues-Xerri Lucile1,Vázquez Ramiro2,Odore Elodie3,Rezai Keyvan3,Kahatt Carmen1,Mackenzie Sarah1,Bekradda Mohamed1,Coudé Marie-Magdelaine4,Dombret Herve4,Gardin Claude4,Lokiec Francois3,Raymond Eric5,Noel Kay6,Cvitkovic Esteban6,Herait Patrice6,Bertoni Francesco2,Riveiro María E.1

Affiliation:

1. Oncology Therapeutic Development, Clichy, France;

2. Institute of Oncology Research, Università della Svizzera Italiana, Bellinzona, Switzerland;

3. RadioPharmacology Department, Curie Institute–Rene Huguenin Hospital, Saint Cloud, France;

4. Laboratoire de Transfert des Leucémies, Université Paris Diderot, Paris, France;

5. Medical Oncology Department, CHUV, Lausanne, Switzerland;

6. Oncoethix SA, Lucerne, Switzerland

Publisher

Informa UK Limited

Subject

Cancer Research,Oncology,Hematology

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