Combination of Sonogashira coupling and 5-endo-dig cyclization for the synthesis of 2,6-disubstituted-5-azaindoles-Reference-Cited by-同舟云学术

Combination of Sonogashira coupling and 5-endo-dig cyclization for the synthesis of 2,6-disubstituted-5-azaindoles

Published:2019-01-16 Issue:3 Volume:49 Page:351-358
ISSN:0039-7911
Container-title:Synthetic Communications
language:en
Short-container-title:Synthetic Communications

Author:

Balfour Michael N.¹,Zukerman-Schpector Julio²,Rodriguez Maria José Dávila²,Reis Joel Savi¹,Esteves Carlos Henrique A.¹,Stefani Hélio A.¹

Affiliation:

1. Faculdade de Ciências Farmacêuticas, Departamento de Farmácia, Universidade de São Paulo, São Paulo, SP, Brazil;

2. Laboratório de Cristalografia, Estereodinâmica e Modelagem Molecular, Departamento de Química, Universidade Federal de São Carlos, São Carlos, SP, Brazil

Funder

São Paulo Research Foundation

Fundação de Amparo a Pesquisa do Estado de São Paulo – FAPESP

National Council for Scientific and Technological Development

Coordination for the Improvement of Higher Education Personnel

CAPES

Publisher

Informa UK Limited

Subject

Organic Chemistry

Link

https://www.tandfonline.com/doi/pdf/10.1080/00397911.2018.1545032

Reference11 articles.

1. Synthesis and benzodiazepine receptor (ω receptor) affinities of 3-substituted derivatives of pyrrolo[2,3-c]pyridine-5-carboxylate, a novel class of ω1 selective ligands1This article is dedicated to the memory of our friend and colleague, Sir Derek Barton.1

2. Synthesis and sar of 2- and 3-substituted 7-azaindoles as potential dopamine D4 ligands

3. Meriolins (3-(Pyrimidin-4-yl)-7-azaindoles): Synthesis, Kinase Inhibitory Activity, Cellular Effects, and Structure of a CDK2/Cyclin A/Meriolin Complex

4. Double Sonogashira reactions on dihalogenated aminopyridines for the assembly of an array of 7-azaindoles bearing triazole and quinoxaline substituents at C-5: Inhibitory bioactivity against Giardia duodenalis trophozoites

5. Structure–activity relationship of antiparasitic and cytotoxic indoloquinoline alkaloids, and their tricyclic and bicyclic analogues

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