Allosteric activation of cytochrome P450 3A4 by efavirenz facilitates midazolam binding-Reference-Cited by-同舟云学术

Allosteric activation of cytochrome P450 3A4 by efavirenz facilitates midazolam binding

Published:2017-12-18 Issue:12 Volume:48 Page:1227-1236
ISSN:0049-8254
Container-title:Xenobiotica
language:en
Short-container-title:Xenobiotica

Author:

Ichikawa Tomohiko¹,Tsujino Hirofumi¹,Miki Takahiro¹,Kobayashi Masaya¹,Matsubara Chiaki¹,Miyata Sara¹,Yamashita Taku²,Takeshita Kohei³,Yonezawa Yasushige⁴,Uno Tadayuki¹

Affiliation:

1. Graduate School of Pharmaceutical Sciences, Osaka University , Suita , Osaka , Japan ,

2. School of Pharmacy and Pharmaceutical Sciences, Mukogawa Women’s University , Nishinomiya , Hyogo , Japan ,

3. Institute for Protein Research, Osaka University , Suita , Osaka , Japan , and

4. High Pressure Protein Research Center, Institute of Advanced Technology, Kindai University , Nishimitani, Kinokawa, Wakayama , Japan

Publisher

Informa UK Limited

Subject

Health, Toxicology and Mutagenesis,Pharmacology,Toxicology,Biochemistry,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/00498254.2017.1412540

Reference58 articles.

1. NON-MICHAELIS-MENTEN KINETICS IN CYTOCHROME P450-CATALYZED REACTIONS

2. A Kinetic, Spectroscopic, and Redox Study of Human Tryptophan 2,3-Dioxygenase

3. Molecular dynamics with coupling to an external bath

4. Heterotropic Activation of the Midazolam Hydroxylase Activity of CYP3A by a Positive Allosteric Modulator of mGlu5: In Vitro to In Vivo Translation and Potential Impact on Clinically Relevant Drug-Drug Interactions

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