Synthesis, biological evaluation and in silico studies of novel thiadiazole-hydrazone derivatives for carbonic anhydrase inhibitory and anticancer activities-Reference-Cited by-同舟云学术

Synthesis, biological evaluation and in silico studies of novel thiadiazole-hydrazone derivatives for carbonic anhydrase inhibitory and anticancer activities

Published:2023-07-03 Issue:7 Volume:34 Page:543-567
ISSN:1062-936X
Container-title:SAR and QSAR in Environmental Research
language:en
Short-container-title:SAR and QSAR in Environmental Research

Author:

Bostancı H.E.¹,Çevik U.A.²,Kapavarapu R.³,Güldiken Y.C.⁴,Inan Z.D.Ş.⁵,Güler Ö.Ö.⁶,Uysal T.K.⁶,Uytun A.²,Çetin F.N.¹,Özkay Y.²,Kaplancıklı Z.A.²

Affiliation:

1. Department of Biochemistry, Faculty of Pharmacy, Cumhuriyet University, Sivas, Turkey

2. Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey

3. Department of Pharmaceutical Chemistry and Phytochemistry, Nirmala College of Pharmacy, Atmakur, India

4. Department of Neurology, Kocaeli University Research and Application Hospital, İzmit, Turkey

5. Department of Histology and Embryology, Sivas Cumhuriyet University, Sivas, Turkey

6. Department of Medical Biology, Faculty of Medicine, Ankara Yildirim Beyazit University, Ankara, Turkey

Funder

reported

Publisher

Informa UK Limited

Subject

Drug Discovery,Molecular Medicine,General Medicine,Bioengineering

Link

https://www.tandfonline.com/doi/pdf/10.1080/1062936X.2023.2240698

Reference39 articles.

1. Synthesis, carbonic anhydrase inhibitory activity, anticancer activity and molecular docking studies of new imidazolyl hydrazone derivatives

2. Synthesis, cytotoxicities, and carbonic anhydrase inhibition activities of pyrazoline–benzenesulfonamide derivatives harboring phenol/polyphenol moieties

3. A combination strategy of structure-based virtual screening, MM-GBSA, cross docking, molecular dynamics and metadynamics simulations used to investigate natural compounds as potent and specific inhibitors of tumor linked human carbonic anhydrase IX

4. Novel 3-(6-methylpyridin-2-yl)coumarin-based chalcones as selective inhibitors of cancer-related carbonic anhydrases IX and XII endowed with anti-proliferative activity

5. Dependence on linkers’ flexibility designed for benzenesulfonamides targeting discovery of novel hCA IX inhibitors as potent anticancer agents

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