Synthesis of novel bis-allyloxy and hydroxypropoxy derivatives of 4, 5-diaryl thiophene-2-carboxylic acid and their biological evaluation
Author:
Publisher
Springer Science and Business Media LLC
Subject
General Chemistry
Link
http://link.springer.com/article/10.1007/s12039-017-1274-6/fulltext.html
Reference30 articles.
1. Reitz D B and Isakson P C 1995 Cyclooxygenase-2 inhibitors Curr. Pharm. Des. 1 211
2. Gadad A K, Palkar M B, Anand K, Noolvi M N, Boreddy T S and Wagwade J 2008 Synthesis and biological evaluation of 2-trifluoromethyl/sulfonamido-5,6-diaryl substituted imidazo[2,1-b]-1,3,4-thiadiazoles: A novel class of cyclooxygenase-2 inhibitors Bioorg. Med. Chem. 16 276
3. Sall D J, Bastian J A, Briggs S L, Buben J A, Chirgadze N Y, Clawson D K, Denney M L, Giera D D, Gifford-Moore D S, Harper R W, Hauser K L, Klimkowski V J, Kohn T J, Lin H-S, McCowan J R, Palkowitz A D, Smith G F, Takeuchi K, Thrasher K J, Tinsley J M, Utterback B G, Yan S-C B and Zhang M 1997 Dibasic Benzo[b]thiophene derivatives as a novel class of active site-directed thrombin inhibitors. 1. Determination of the serine protease selectivity, structure–activity relationships, and binding orientation J. Med. Chem. 40 3489
4. Leblanc Y, Roy P, Boyce S, Brideau C, Chan C C, Charleson S, Gordon R, Grimm E, Guay J, Léger S, Li C S, Riendeau D, Visco D, Wang Z, Webb J, Xu L J and Prasit P 1999 SAR in the alkoxy lactone series: The discovery of DFP, a potent and orally active COX-2 inhibitor Bioorg. Med. Chem. Lett. 9 2207
5. Lau C K, Brideau C, Chi Chung C, Charleson S, Cromlish W A, Ethier D, Gauthier J Y, Gordon R, Guay J, Kargman S, Li C-S, Prasit P, Reindeau D, Thérien M, Visco D M and Lijing X 1999 Synthesis and biological evaluation of 3-heteroaryloxy-4-phenyl-2(5H)- furanones as selective COX-2 inhibitors Bioorg. Med. Chem. Lett. 9 3187
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