Idalopirdine – a small molecule antagonist of 5-HT6 with therapeutic potential against obesity-Reference-Cited by-同舟云学术

Idalopirdine – a small molecule antagonist of 5-HT6 with therapeutic potential against obesity

Published:2015-09-29 Issue:6 Volume:30 Page:1487-1494
ISSN:0885-7490
Container-title:Metabolic Brain Disease
language:en
Short-container-title:Metab Brain Dis

Author:

Dudek Magdalena,Marcinkowska Monika,Bucki Adam,Olczyk Adrian,Kołaczkowski Marcin

Publisher

Springer Science and Business Media LLC

Subject

Cellular and Molecular Neuroscience,Clinical Neurology,Biochemistry

Link

http://link.springer.com/content/pdf/10.1007/s11011-015-9736-3.pdf

Reference27 articles.

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2. Brown M, Bing C, King P, Pickavance L, Heal D, Wilding J (2001) Sibutramine reduces feeding, body fat and improves insulin resistance in dietary-obese male Wistar rats independently of hypothalamic neuropeptide Y. Br J Pharmacol 132:1898–1904

3. Caldirola P (2003) 5-HT6 receptor antagonism. A novel mechanism for the management of obesity. SMI Inaugural Conference on Obesity and Related Disorders, London

4. Choi S, Blake V, Cole S, Fernstrom JD (2006) Effects of chronic fenfluramine administration on hypothalamic neuropeptide mRNA expression. Brain Res 1087:83–86

5. Clissold KA, Choi E, Pratt WE (2013) Serotonin 1A, 1B and 7 receptors of the rat medial nucleus accumbens differentially regulate feeding, water intake, and locomotor activity. Pharmacol Biochem Behav 112:1–17

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