In vitro identification of the cytochrome P450 isozymes involved in the N-demethylation of the active opioid metabolite nortilidine to bisnortilidine

Author:

Wustrow Isabel,Riedel Klaus-Dieter,Mikus Gerd,Weiss Johanna

Publisher

Springer Science and Business Media LLC

Subject

Pharmacology,General Medicine

Reference19 articles.

1. Grün B, Krautter S, Riedel K-D, Mikus G (2009) Inhibition of the active principle of the weak opioid tilidine by the triazole antifungal voriconazole. Br J Clin Pharmacol 68:712–720

2. Hajda JP, Jahnchen E, Oie S, Trenk D (2002) Sequential first-pass metabolism of nortilidine: the active metabolite of the synthetic opioid drug tilidine. J Clin Pharmacol 42:1257–1261

3. Hesse LM, von Moltke LL, Shader RI, Greenblatt DJ (2001) Ritonavir, efavirenz, and nelfinavir inhibit CYP2B6 activity in vitro: potential drug interactions with bupropion. Drug Metab Dispos 29:100–102

4. International Narcotics Board Control (INCB) (2011) Estimated world requirements of narcotic drugs in grams for 2011. http://www.incb.org/pdf/e/estim/2011/EstFeb11.pdf . Accessed 05 Feb 2011

5. Obach RS (1997) Nonspecific binding to microsomes: impact on scale-up of in vitro intrinsic clearance to hepatic clearance as assessed through examination of warfarin, imipramine, and propranolol. Drug Metab Dispos 25:1359–1369

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