SMART Drug Design: Novel Phosphopeptide and ATP Mimetic-Based Small Molecule Inhibitors of the Oncogenic Protein Kinase pp60src (Src)
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Publisher
Springer US
Link
http://link.springer.com/content/pdf/10.1007/0-387-24532-4_11
Reference185 articles.
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3. Alfaro-Lopez, J., Yuan, W., Phan, B.C., Kamath, J., Lou, Q., Lam, K.S., and Hruby, V.J. (1998). Discovery of a novel series of potent and selective substrate-based inhibitors of pp60c-src protein tyrosine kinase: conformational and topographical constraints in peptide design. J. Med. Chem. 41:2252–2260.
4. Alligood, K.J., Charifson, P.S., Crosby, R., Consler, T.G., Feldman, P.L., Gampe, R.T. Jr., Gilmer, T.M., Jordan, S.R., Milstead, M.W., Mohr, C., Peel, M.R., Rocque, W., Rodriguez, M., Rusnak, D.W., Shewchuk, L.M., and Sternbach, D.D. (1998). The formation of a covalent complex between a dipeptide ligand and the SRC SH2 domain. Bioorg. Med. Chem. Lett. 8:1189–1194.
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Cited by 2 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Novel Small-Molecule Inhibitors of Src Kinase for Cancer Therapy;Topics in Medicinal Chemistry;2007
2. Protein Kinases and Protein Phosphatases in Signal Transduction Pathways;Comprehensive Medicinal Chemistry II;2007
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