Exploring 1-adamantanamine as an alternative amine moiety for metabolically labile azepane ring in newly synthesized benzo[d]thiazol-2(3H)one σ receptor ligands-Reference-Cited by-同舟云学术

Exploring 1-adamantanamine as an alternative amine moiety for metabolically labile azepane ring in newly synthesized benzo[d]thiazol-2(3H)one σ receptor ligands

Published:2020-07-08 Issue:9 Volume:29 Page:1697-1706
ISSN:1054-2523
Container-title:Medicinal Chemistry Research
language:en
Short-container-title:Med Chem Res

Author:

Intagliata Sebastiano,Agha Hebaalla,Kopajtic Theresa A.,Katz Jonathan L.,Kamble Shyam H.,Sharma Abhisheak,Avery Bonnie A.,McCurdy Christopher R.

Publisher

Springer Science and Business Media LLC

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics

Link

http://link.springer.com/content/pdf/10.1007/s00044-020-02597-2.pdf

Reference45 articles.

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2. Avery BA, Vuppala PK, Jamalapuram S, Sharma A, Mesangeau C, Chin FT, McCurdy CR (2017) Quantification of highly selective sigma-1 receptor antagonist CM304 using liquid chromatography tandem mass spectrometry and its application to a pre-clinical pharmacokinetic study. Drug Test Anal 9(8):1236–1242. https://doi.org/10.1002/dta.2156

3. Bangaru ML, Weihrauch D, Tang QB, Zoga V, Hogan Q, Wu HE (2013) Sigma-1 receptor expression in sensory neurons and the effect of painful peripheral nerve injury. Mol Pain 9:47. https://doi.org/10.1186/1744-8069-9-47

4. Bhat R, Fishback JA, Matsumoto RR, Poupaert JH, McCurdy CR (2013) Structure activity relationship study of benzo[d]thiazol-2(3H)one based sigma receptor ligands. Bioorg Med Chem Lett 23(17):5011–5013. https://doi.org/10.1016/j.bmcl.2013.06.032

5. Bowen WD, DeCosta BR, Hellewell SB, Walker JM, Rice KC (1993) [3H]-(+)-Pentazocine: a potent and highly selective benzomorphan-based probe for sigma-1 receptors. Mol Neuropharmacol 3:117–126

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