Design, synthesis and cytotoxicity evaluation of pyrazolyl pyrazoline and pyrazolyl aminopyrimidine derivatives as potential anticancer agents
Author:
Publisher
Springer Science and Business Media LLC
Subject
Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics
Link
http://link.springer.com/article/10.1007/s00044-017-2082-8/fulltext.html
Reference41 articles.
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2. Acker TM, Khatri A, Vance KM, Slabber C, Bacsa J, Snyder JP, Traynelis SF, Liotta DC (2013) Structure-activity relationships and pharmacophore model of a noncompetitive pyrazoline containing class of GluN2C/GluN2D selective antagonists. J Med Chem 56:6434–6456
3. Alam R, Alam MA, Panda AK, Rahisuddin (2016a) Design, synthesis and cytotoxicity evaluation of novel (E)-3-(3-aryl-1-phenyl-1H-pyrazol-4-yl)-1-(pyridin-3-yl)prop-2-en-1-ones as anticancer agents. Heterocycl Commun 22:221–225
4. Alam R, Alam MA, Panda AK, Rahisuddin (2017) Design, synthesis and cytotoxicity evaluation of 3-(5-(3-(aryl)-1-phenyl-1H-pyrazol-4-yl)-1-phenyl-4,5-dihydro-1H-pyrazol-3-yl)pyridine and 5-(3-(aryl)-1-phenyl-1h-pyrazol-4-yl)-3-(pyridin-3-yl)-4,5-dihydropyrazole-1-carbaldehyde derivatives as potential anticancer agents. J Heterocycl Chem 54:1812–1821
5. Alam R, Wahi D, Singh R, Sinha D, Tandon V, Grover A, Rahisuddin (2016b) Design, synthesis, cytotoxicity, human topoisomerase iiα inhibitory activity and molecular docking studies of pyrazole derivatives as potential anticancer agents. Bioorg Chem 69:77–90
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