Hologram quantative structure–activity relationship studies on 1-(5-carboxyindol-1-yl)propan-2-one inhibitors of human cytosolic phospholipase A2α
Author:
Publisher
Springer Science and Business Media LLC
Subject
Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics
Link
http://link.springer.com/content/pdf/10.1007/s00044-013-0763-5.pdf
Reference25 articles.
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3. Chen L, Wang W, Lee KL, Shen MWH, Murphy EA, Zhang W, Xu X, Tam S, Nickerson-Nutter C, Goodwin DG, Clark JD, McKew JC (2009) Reactions of functionalized sulfonamides: application to lowering the lipophilicity of cytosolic phospholipase Α2α inhibitors. J Med Chem 52(4):1156–1171. doi: 10.1021/jm8009876
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5. Connolly S, Robinson DH (1995) Patent update: pulmonary-allergy, dermatological, gastrointestinal and arthritis: the search for inhibitors of the phospholipases A2. Expert Opin Ther Pat 5(7):673–683. doi: 10.1517/13543776.5.7.673
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