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Cytotoxic activities and metabolic studies of new combretastatin analogues

  • Published:2015-04-09 Issue:8 Volume:24 Page:3143-3156
  • ISSN:1054-2523
  • Container-title:Medicinal Chemistry Research
  • language:en
  • Short-container-title:Med Chem Res

Author:

Macé Yohan,Bony Emilie,Delvaux David,Pinto Adan,Mathieu Véronique,Kiss Robert,Feron Olivier,Quetin-Leclercq Joëlle,Riant Olivier

Publisher

Springer Science and Business Media LLC

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics

Reference26 articles.

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2. Aguirre G, Boiani L, Boiani M, Cerecetto H, Di Maio R, Gonzalez M, Porcal W, Denicola A, Piro OE, Castellano EE, Sant’Anna CMR, Barreiro EJ (2005) New potent 5-substituted benzofuroxans as inhibitors of Trypanosoma cruzi growth: quantitative structure–activity relationship studies. Bioorg Med Chem 13:6336–6346

3. Bedford SB, Quarterman CP, Rathbone DL, Slack JA, Griffin RJ, Stevens MFG (1996) Synthesis of water-soluble prodrugs of the cytotoxic agent combretastatin A4. Bioorg Med Chem Lett 6:157–160

4. Boiani M, Boiani L, Denicola A, Torres de Ortiz S, Serna E, Vera de Bilbao N, Sanabria L, Yaluff G, Nakayama H, Rojas de Arias A, Vega C, Rolan M, Gomez-Barrio A, Cerecetto H, Gonzalez M (2006) 2H-benzimidazole 1,3-dioxide derivatives: a new family of water-soluble anti-trypanosomatid agents. J Med Chem 49:3215–3224

5. Carroll WA, Altenbach RJ, Bai H, Brioni JD, Brune ME, Buckner SA, Cassidy C, Chen Y, Coghlan MJ, Daza AV, Drizin I, Fey TA, Fitzgerald M, Gopalakrishnan M, Gregg RJ, Henry RF, Holladay MW, King LL, Kort ME, Kym PR, Milicic I, Tang R, Turner SC, Whiteaker KL, Yi L, Zhang H, Sullivan JP (2004) Synthesis and structure–activity relationships of a novel series of 2,3,5,6,7,9-hexahydrothieno[3,2-b]quinolin-8(4H)-one 1,1-dioxide K(ATP) channel openers: discovery of (-)-(9S)-9-(3-bromo-4-fluorophenyl)-2,3,5,6,7,9-hexahydrothieno[3,2-b]quinolin-8(4H)-one 1,1-dioxide (A-278637), a potent K(ATP) opener that selectively inhibits spontaneous bladder contractions. J Med Chem 47:3163–3179
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