Exploring thiazole-linked thioureas using alkaline phosphatase assay, biochemical evaluation, computational analysis and structure–activity relationship (SAR) studies-Reference-Cited by-同舟云学术

Exploring thiazole-linked thioureas using alkaline phosphatase assay, biochemical evaluation, computational analysis and structure–activity relationship (SAR) studies

Published:2022-08-13 Issue:10 Volume:31 Page:1792-1802
ISSN:1054-2523
Container-title:Medicinal Chemistry Research
language:en
Short-container-title:Med Chem Res

Author:

Channar Sajid Ali,Channar Pervaiz Ali,Saeed Aamer,Alsfouk Aisha A.,Ejaz Syeda Abida^ORCID,Ujan Rabail,Noor Razia,Bilal Muhammad Sajjad,Abbas Qamar,Hussain Zahid,Khan Bilal Ahmad,Raza Hussain,Indher Hafiz Abdul Bari,Mahesar Parvez Ali

Publisher

Springer Science and Business Media LLC

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics

Link

https://link.springer.com/content/pdf/10.1007/s00044-022-02945-4.pdf

Reference40 articles.

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3. Bell FW, Cantrell AS, Hoegberg M, Jaskunas SR, Johansson NG, Jorden CL, et al. Phenethylthiazolethiourea (PETT) compounds, a new class of HIV-1 reverse transcriptase inhibitors. 1. Synthesis and basic structure–activity relationship studies of PETT analogs. J Med Chem. 1995;38:4929–36.

4. Patt WC, Hamilton HW, Taylor MD, Ryan MJ, Taylor DG Jr, Connoly CJC, et al. Structure–activity relationships of a series of 2-amino-4-thiazole-containing renin inhibitors. J Med Chem. 1992;35:2562–72.

5. Tsuji K, Ishikawa H. Synthesis and anti-pseudomonal activity of new 2-isocephems with a dihydroxypyridone moiety at C-7. Bioorg Med Chem Lett. 1994;4:1601–6.

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