Design, synthesis, and <i>in vitro</i> and <i>in silico</i> studies of morpholine derived thiazoles as bovine carbonic anhydrase-II inhibitors-Reference-Cited by-同舟云学术

Design, synthesis, and in vitro and in silico studies of morpholine derived thiazoles as bovine carbonic anhydrase-II inhibitors

Published:2024 Issue:30 Volume:14 Page:21355-21374
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Tasleem Mussarat¹^ORCID,Ullah Saeed²,Khan Ajmal²,Mali Suraj N.³^ORCID,Kumar Sunil⁴,Mathew Bijo⁴,Oneto Angelo⁵,Noreen Faiqa¹,Eldesoky Gaber E.⁶,Schenone Silvia⁷,Al-Harrasi Ahmed²,Shafiq Zahid¹⁵^ORCID

Affiliation:

1. Institute of Chemical Sciences, Bahauddin Zakariya University, Multan-60800, Pakistan

2. Natural and Medical Sciences Research Centre, University of Nizwa, P.O. Box 33, PC 616, Birkat Al Mauz, Nizwa, Sultanate of Oman

3. School of Pharmacy, D. Y. Patil University (Deemed to be University), Sector 7, Nerul, Navi Mumbai 400706, India

4. Department of Pharmaceutical Chemistry, Amrita School of Pharmacy, Amrita Vishwa Vidyapeetham, AIMS Health Sciences Campus, Kochi 682041, India

5. Department of Pharmaceutical & Medicinal Chemistry, An der Immenburg 4, D-53121 Bonn, Germany

6. Chemistry Department, College of Science, King Saud University, Riyadh 11451, Saudi Arabia

7. Department of Pharmacy, University of Genoa, Viale Benedetto XV, 3, Genoa 16132, Italy

Abstract

Morpholine based thiazoles have been reported as bovine carbonic anhydrase CA-II inhibitors.

Funder

King Saud University

Alexander von Humboldt-Stiftung

Publisher

Royal Society of Chemistry (RSC)

Link

http://pubs.rsc.org/en/content/articlepdf/2024/RA/D4RA03385J

Reference40 articles.

1. Quinazolinones as Competitive Inhibitors of Carbonic Anhydrase-II (Human and Bovine): Synthesis, in-vitro, in-silico, Selectivity, and Kinetics Studies

2. Carbonic anhydrase inhibitors

3. Emerging role of carbonic anhydrase inhibitors

4. Novel carbonic anhydrase inhibitors

5. Structure–activity relationships for the interaction of 5,10-dihydroindeno[1,2-b]indole derivatives with human and bovine carbonic anhydrase isoforms I, II, III, IV and VI