Drug interactions with Bruton’s tyrosine kinase inhibitors: clinical implications and management

Author:

Fancher Karen M.ORCID,Pappacena Jeremy J.

Publisher

Springer Science and Business Media LLC

Subject

Pharmacology (medical),Cancer Research,Pharmacology,Toxicology,Oncology

Reference45 articles.

1. Roskoski R (2016) Ibrutinib inhibition of Bruton protein-tyrosine kinase (BTK) in the treatment of B cell neoplasms. Pharmacol Res 113(Pt A):395–408

2. Barf T, Covey T, Izumi R et al (2017) Acalabrutinib (ACP-196): a covalent bruton tyrosine kinase inhibitor with a differentiated selectivity and in vivo potency profile. J Pharmacol Exp Ther 363:240–252

3. (2018) Imbruvica® (ibrutinib) [package insert]. Janssen Biotech, Inc., Horsham, PA

4. (2019) Calquence® (acalabrutinib) [package insert]. AstraZeneca Pharmaceuticals LP, Wilmington, DE

5. (2019) Brukinsa® (zanubrutinib) [package insert]. BeiGene USA, Inc., San Mateo, CA

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